INN name:
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Tazemetostat
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Lab codes:
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E-7438, EPZ-6438
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Chemical name:
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N-[(4,6-dimethyl-2-oxo-1,2-dihydropyridin-3-yl)methyl]-5-[ethyl(oxan-4-yl)amino]-4-methyl-4'-[(morpholin-4-yl)methyl][1,1'-biphenyl]-3-carboxamide
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Molecular formula:
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C34H44N4O4
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Chemical Structure:
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CAS Registry Number:
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1403254-99-8
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Originator:
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Epizyme
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Class:
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Antineoplastic
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Mechanism of Action:
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EZH2 enzyme
inhibitors
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WHO ATC code:
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L01X-X
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EPhMRA code:
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L1X9
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Clinical Trials:
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Thursday, 17 September 2015
Tazemetostat
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