INN name:
|
Erdafitinib
|
Lab codes:
|
JNJ-42756493
|
Chemical name:
|
N1-(3,5-dimethoxyphenyl)-N1-[3-(1-methyl-1H-pyrazol-4-yl)quinoxalin-6-yl]-N2-(propan-2-yl)ethane-1,2-diamine
|
Molecular formula:
|
C25H30N6O2
|
Chemical Structure:
|
 |
CAS Registry Number:
|
1346242-81-6
|
Originator:
|
Astex
Therapeutics
|
Developer:
|
Janssen
Research & Development
|
Class:
|
Antineoplastics
|
Mechanism of Action:
|
Fibroblast
growth factor receptor antagonists
|
WHO ATC code:
|
L01
(Antineoplastic Agents)
|
EPhMRA code:
|
L1
(Antineoplastics)
|
Clinical Trials:
Conditions
|
Phases
|
Status
|
Urothelial
Cancer
|
Phase
2
|
Recruiting
|
Tumor
or Lymphoma
|
Phase
1
|
Recruiting
|
Neoplasms; Lymphoma;
Adenocarcinoma; Esophagogastric Junction
|
Phase
1
|
Recruiting
|
Carcinoma, Hepatocellular
|
Phase
1
|
Recruiting
|
|
|
|
Recent activities on the
drug:
|
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