Thursday 17 September 2015

Tazemetostat

INN name:

Tazemetostat
Lab codes:

E-7438, EPZ-6438
Chemical name:

N-[(4,6-dimethyl-2-oxo-1,2-dihydropyridin-3-yl)methyl]-5-[ethyl(oxan-4-yl)amino]-4-methyl-4'-[(morpholin-4-yl)methyl][1,1'-biphenyl]-3-carboxamide

Molecular formula:

C34H44N4O4
Chemical Structure:


CAS Registry Number:

1403254-99-8
Originator:

Epizyme
Class:

Antineoplastic
Mechanism of Action:

EZH2 enzyme inhibitors
WHO ATC code:

L01X-X
EPhMRA code:

L1X9

Clinical Trials:

Indication
Phase
Status
Follicular Lymphoma
Phase 2
Recruiting
Diffuse Large B-cell Lymphoma
Phase 2
Recruiting
Advanced Solid Tumors
Phase 1
Recruiting
B-cell Lymphoma
Phase 1
Recruiting

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