Thursday 17 September 2015

Pinometostat

INN name:

Pinometostat
Lab codes:

EPZ-5676
Chemical name:

9-{5-deoxy-5-[{cis-3-[2-(5-tert-butyl-1H-benzimidazol-2-yl)ethyl]cyclobutyl}(propan-2-yl)amino]-beta-D-ribofuranosyl}-9H-purin-6-amine

Molecular formula:

C30H42N8O3
Chemical Structure:


CAS Registry Number:

1380288-87-8
Originator:

Epizyme
Class:

Antineoplastic
Mechanism of Action:

DOT1L protein inhibitors
WHO ATC code:

L01X-X
EPhMRA code:

L1X

Clinical Trials:

Indication
Phase
Intervention
Status
Leukemia
Phase 1
Alone
Recruiting




Recent activities on the drug:

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