Thursday 17 September 2015

Spebrutinib

INN name:

Spebrutinib
Lab codes:

AVL-292, CC-292
Chemical name:

N-[3-({5-fluoro-2-[4-(2-methoxyethoxy)anilino]pyrimidin-4-yl}amino)phenyl]prop-2-enamide

Molecular formula:

C22H22FN5O3
Chemical Structure:

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CAS Registry Number:

1202757-89-8
Originator:

Avila Therapeutics
Developer:

Celgene Corporation
Class:

Antineoplastic
Mechanism of Action:

Tyrosine kinase inhibitor
WHO ATC code:

L01X-E (Protein kinase inhibitors)
M01A (Antiinflammatory and Antirheumatic Products, Non-steroids)

EPhMRA code:

L1H (Protein Kinase Inhibitor Antineoplastics)
M1A (Anti-Rheumatics, Non-Steroidal)

Clinical Trials:

Conditions
Phases
Interventions
Status
Rheumatoid Arthritis
Phase 2
Alone
Recruiting
Lymphoma, Large B-Cell, Diffuse
Phase 1
Combination
Recruiting
Relapsed/Refractory B-cell Lymphoma
Phase 1
Combination
Active, not recruiting
Healthy Volunteers
Phase 1
Combination
Completed
Leukemia Lymphocytic Chronic B-Cell
Phase 1
Combination
Active, not recruiting
Leukemia Lymphocytic Chronic B-Cell
Phase 1
Combination
Active, not recruiting
B Cell Non-Hodgkin's Lymphoma|Chronic Lymphocytic Leukemia|Waldenstrom Macroglobulinemia
Phase 1
Alone
Completed




Recent activities on the drug:

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