Thursday 17 September 2015

Infigratinib

INN name:

Infigratinib
Lab codes:

BGJ-398; NVP-BGJ398
Chemical name:

N'-(2,6-dichloro-3,5-dimethoxyphenyl)-N-{6-[4-(4-ethylpiperazin-1-yl)anilino]pyrimidin-4-yl}-N-methylurea

Molecular formula:

C26H31Cl2N7O3
Chemical Structure:

Add caption

CAS Registry Number:

872511-34-7
Originator:

Novartis
Class:

Antineoplastics
Mechanism of Action:

Tyrosine kinase inhibitor
WHO ATC code:

L01X-E
EPhMRA code:

L1H

Clinical Trials:

Conditions
Phases
Interventions
Status
Advanced Cholangiocarcinoma
Phase 2
Alone
Recruiting
Melanoma
Phase 2
Combination
Active, not recruiting
Melanoma
Phase 2
Combination
Recruiting
Recurrent Glioblastoma or Other Glioma Subtypes
Phase 2
Alone
Recruiting
Solid Tumor|Hematologic Malignancies
Phase 2
Alone
Recruiting
Advanced Gastrointestinal Stromal Tumor (GIST)
Phase 1|Phase 2
Combination
Recruiting
Advanced Solid Malignancies
Phase 1
Alone
Recruiting
Advanced Solid Tumors,|Metastatic Solid Tumors
Phase 1
Combination
Recruiting
Cancer of Cervix|Tumors
Phase 1
Combination
Withdrawn
Tumor With Alterations of the FGF-R
Phase 1
Alone
Recruiting


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